P4532-50MG Display Image

(-)-N6-(2-Phenylisopropyl)adenosine, solid

Code: P4532-50MG D2-231

Biochem/physiol Actions

A1 adenosine receptor agonist. Affinity for adenosine receptor is approx. 100× that of the (+)-isomer.

Features and Bene...


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Your Price
£219.00 50MG
£262.80 inc. VAT

Biochem/physiol Actions

A1 adenosine receptor agonist. Affinity for adenosine receptor is approx. 100× that of the (+)-isomer.

Features and Benefits

This compound is featured on the Adenosine Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here.

Packaging

50, 100 mg in glass bottle

25 mg in poly bottle

colorwhite
formsolid
Gene Informationhuman ... ADORA1(134)
InChI keyRIRGCFBBHQEQQH-SSFGXONLSA-N
InChI1S/C19H23N5O4/c1-11(7-12-5-3-2-4-6-12)23-17-14-18(21-9-20-17)24(10-22-14)19-16(27)15(26)13(8-25)28-19/h2-6,9-11,13,15-16,19,25-27H,7-8H2,1H3,(H,20,21,23)/t11-,13-,15-,16-,19-/m1/s1
potency1.17 nM Ki for A1 receptors (using [3H]CHA in rat forebrain preparations)
Quality Level200
SMILES stringC[C@H](Cc1ccccc1)Nc2ncnc3n(cnc23)[C@@H]4O[C@H](CO)[C@@H](O)[C@H]4O
solubilityH2O: slightly soluble 0.3 mg/mL (Solutions may be stored for several days at 4°C.), 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: 1.6 mg/mL (Solutions may be stored for several days at 4°C.)
storage temp.2-8°C
Code
Description
Unit Size
List Price
Qty
P4532-25MG
Unit:25MG
List Price: £118.00
Source:List Price
ADD
Cas Number38594-96-6
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